Positive allosteric modulators of the α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor

J Med Chem. 2010 Oct 28;53(20):7271-9. doi: 10.1021/jm1000419.
No abstract available

MeSH terms

  • Allosteric Regulation
  • Animals
  • Benzamides / chemistry
  • Benzamides / pharmacology
  • Benzothiadiazines / chemistry
  • Benzothiadiazines / pharmacology
  • Binding Sites
  • Excitatory Amino Acid Agents / chemistry*
  • Excitatory Amino Acid Agents / pharmacology
  • Humans
  • Indazoles / chemistry
  • Indazoles / pharmacology
  • Ligands
  • Models, Molecular
  • Protein Conformation
  • Receptors, AMPA / chemistry
  • Receptors, AMPA / physiology*
  • Sulfonamides / chemistry
  • Sulfonamides / pharmacology

Substances

  • Benzamides
  • Benzothiadiazines
  • Excitatory Amino Acid Agents
  • Indazoles
  • Ligands
  • Receptors, AMPA
  • Sulfonamides